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Assay Detail

CHEMBL4021271

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Functional
Cytotoxicity against mouse LMM3 cells
4
Total Activities
4
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Organism Mus musculus
Cell Type LMM3
Confidence 1 — Organism
Curated By Autocuration

Target

LMM3 cell line (CHEMBL614095)
Type CELL-LINE
Organism Mus musculus

Publication

Indoles as therapeutics of interest in medicinal chemistry: Bird's eye view.
Chadha N, Silakari O.
Eur J Med Chem (2017) 134 : 159 -184
PubMed 28412530 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 4 4.85 5.03

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL44541 MERIDIANIN C 1 5.03
CHEMBL296682 MERIDIANIN E 1 4.96
CHEMBL44545 MERIDIANIN B 1 4.94
CHEMBL46440 MERIDIANIN D 1 4.47

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL44541 MERIDIANIN C IC50 = 9300.0 nM 5.03
CHEMBL296682 MERIDIANIN E IC50 = 11100.0 nM 4.96
CHEMBL44545 MERIDIANIN B IC50 = 11400.0 nM 4.94
CHEMBL46440 MERIDIANIN D IC50 = 33900.0 nM 4.47