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Assay Detail

CHEMBL4022854

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Binding
Inhibition of wild type C57BL/6 mouse small intestinal sucrase/isomaltase using sucrose as substrate after 30 mins
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Binding
Organism Mus musculus
Confidence 9 — Direct single protein target
Curated By Autocuration

Target

Sucrase-isomaltase (CHEMBL1667666)
Type SINGLE PROTEIN
Organism Mus musculus

Publication

N-Butyl-l-deoxynojirimycin (l-NBDNJ): Synthesis of an Allosteric Enhancer of α-Glucosidase Activity for the Treatment of Pompe Disease.
D'Alonzo D, De Fenza M, Porto C, Iacono R, Huebecker M, Cobucci-Ponzano B, Priestman DA, Platt F, Parenti G, Moracci M, Palumbo G, Guaragna A.
J Med Chem (2017) 60 : 9462 -9469
PubMed 29112434 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 2 5.82 5.82

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL1029 MIGLUSTAT 4.0 1 5.82
CHEMBL4061367 1 -

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL1029 MIGLUSTAT IC50 = 1500.0 nM 5.82
CHEMBL4061367 IC50 = 2000000.0 nM -