Skip to main content
Free research Free research Free assay review with research home and workspace preview
Quick search ChEMBL 36
Assay Detail

CHEMBL4026907

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Binding
Binding affinity to GST (unknown origin) by fluorescence polarization assay
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Binding
Organism Homo sapiens
Confidence 0 — Uncurated / Unknown
Curated By Autocuration

Target

Unchecked (CHEMBL612545)
Type UNCHECKED

Publication

One-Bead-Two-Compound Thioether Bridged Macrocyclic γ-AApeptide Screening Library against EphA2.
Shi Y, Challa S, Sang P, She F, Li C, Gray GM, Nimmagadda A, Teng P, Odom T, Wang Y, van der Vaart A, Li Q, Cai J.
J Med Chem (2017) 60 : 9290 -9298
PubMed 29111705 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
Kd 1 4.85 4.85

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL4071045 1 4.85

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL4071045 Kd = 14200.0 nM 4.85