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Assay Detail

CHEMBL4029426

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Functional
Induction of proton motive force collapse in Escherichia coli inverted membrane vesicle in presence of ATP-driven PMF generation system by ACMA-based fluorescence assay
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Organism Escherichia coli
Confidence 0 — Uncurated / Unknown
Curated By Autocuration

Target

Unchecked (CHEMBL612545)
Type UNCHECKED

Publication

Phenylthiazole Antibacterial Agents Targeting Cell Wall Synthesis Exhibit Potent Activity in Vitro and in Vivo against Vancomycin-Resistant Enterococci.
Mohammad H, Younis W, Chen L, Peters CE, Pogliano J, Pogliano K, Cooper B, Zhang J, Mayhoub A, Oldfield E, Cushman M, Seleem MN.
J Med Chem (2017) 60 : 2425 -2438
PubMed 28248504 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
EC50 2 5.66 6.40

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL224214 CARBONYL CYANIDE M-CHLOROPHENYLHYDRAZONE 1 6.40
CHEMBL1798027 1 4.92

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL224214 CARBONYL CYANIDE M-CHLOROPHENYLHYDRAZONE EC50 = 400.0 nM 6.40
CHEMBL1798027 EC50 = 12000.0 nM 4.92