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Assay Detail

CHEMBL4031916

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Functional
Agonist activity at recombinant mouse OTR expressed in CHO-K1 cells assessed as induction of Ca2+ mobilization after overnight incubation by FLIPR assay
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Organism Mus musculus
Confidence 9 — Direct single protein target
Curated By Autocuration

Target

Oxytocin receptor (CHEMBL3243907)
Type SINGLE PROTEIN
Organism Mus musculus

Publication

Targets for Drug Therapy for Autism Spectrum Disorder: Challenges and Future Directions.
Lacivita E, Perrone R, Margari L, Leopoldo M.
J Med Chem (2017) 60 : 9114 -9141
PubMed 29039668 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
EC50 1 7.54 7.54

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL3763342 1 7.54

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL3763342 EC50 = 29.0 nM 7.54