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Assay Detail

CHEMBL4032330

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Binding
Inhibition of human liver LDHA using sodium pyruvate as substrate after 5 mins in presence of NAPDH and EDTA by diaphorase/resazurin based fluorescence assay
67
Total Activities
67
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Binding
Organism Homo sapiens
Confidence 9 — Direct single protein target
Curated By Autocuration

Target

L-lactate dehydrogenase A chain (CHEMBL4835)
Type SINGLE PROTEIN
Organism Homo sapiens

Publication

Discovery and Optimization of Potent, Cell-Active Pyrazole-Based Inhibitors of Lactate Dehydrogenase (LDH).
Rai G, Brimacombe KR, Mott BT, Urban DJ, Hu X, Yang SM, Lee TD, Cheff DM, Kouznetsova J, Benavides GA, Pohida K, Kuenstner EJ, Luci DK, Lukacs CM, Davies DR, Dranow DM, Zhu H, Sulikowski G, Moore WJ, Stott GM, Flint AJ, Hall MD, Darley-Usmar VM, Neckers LM, Dang CV, Waterson AG, Simeonov A, Jadhav A, Maloney DJ.
J Med Chem (2017) 60 : 9184 -9204
PubMed 29120638 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 67 6.38 8.05

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL4059985 1 8.05
CHEMBL4090677 1 7.72
CHEMBL4100845 1 7.57
CHEMBL4081890 1 7.50
CHEMBL3335794 1 7.42
CHEMBL4080497 1 7.42
CHEMBL4069726 1 7.38
CHEMBL4101800 1 7.28
CHEMBL4076027 1 7.24
CHEMBL4075666 1 7.19
CHEMBL4062709 1 7.19
CHEMBL4076958 1 7.04
CHEMBL4069796 1 7.02
CHEMBL4082867 1 6.96
CHEMBL4067976 1 6.94
CHEMBL4098516 1 6.91
CHEMBL4095368 1 6.86
CHEMBL4090794 1 6.75
CHEMBL4063125 1 6.46
CHEMBL4066429 1 6.46
CHEMBL4065858 1 6.37
CHEMBL4076973 1 6.17
CHEMBL4099443 1 6.12
CHEMBL2059811 1 5.87
CHEMBL4084774 1 5.62
CHEMBL4092360 1 5.21
CHEMBL4079793 1 4.76
CHEMBL4079457 1 4.59
CHEMBL4077586 1 4.56
CHEMBL4098402 1 4.56

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL4059985 IC50 = 9.0 nM 8.05
CHEMBL4090677 IC50 = 19.0 nM 7.72
CHEMBL4100845 IC50 = 27.0 nM 7.57
CHEMBL4081890 IC50 = 32.0 nM 7.50
CHEMBL3335794 IC50 = 38.0 nM 7.42
CHEMBL4080497 IC50 = 38.0 nM 7.42
CHEMBL4069726 IC50 = 42.0 nM 7.38
CHEMBL4101800 IC50 = 53.0 nM 7.28
CHEMBL4076027 IC50 = 57.0 nM 7.24
CHEMBL4075666 IC50 = 65.0 nM 7.19
CHEMBL4062709 IC50 = 65.0 nM 7.19
CHEMBL4076958 IC50 = 91.0 nM 7.04
CHEMBL4069796 IC50 = 95.0 nM 7.02
CHEMBL4082867 IC50 = 110.0 nM 6.96
CHEMBL4067976 IC50 = 115.0 nM 6.94
CHEMBL4098516 IC50 = 124.0 nM 6.91
CHEMBL4095368 IC50 = 139.0 nM 6.86
CHEMBL4090794 IC50 = 176.0 nM 6.75
CHEMBL4063125 IC50 = 349.0 nM 6.46
CHEMBL4066429 IC50 = 349.0 nM 6.46
CHEMBL4065858 IC50 = 424.0 nM 6.37
CHEMBL4076973 IC50 = 672.0 nM 6.17
CHEMBL4099443 IC50 = 754.0 nM 6.12
CHEMBL2059811 IC50 = 1340.0 nM 5.87
CHEMBL4084774 IC50 = 2370.0 nM 5.62
CHEMBL4092360 IC50 = 6230.0 nM 5.21
CHEMBL4079793 IC50 = 17300.0 nM 4.76
CHEMBL4079457 IC50 = 25500.0 nM 4.59
CHEMBL4077586 IC50 = 27700.0 nM 4.56
CHEMBL4098402 IC50 = 27700.0 nM 4.56
CHEMBL1479261 IC50 = 28800.0 nM 4.54
CHEMBL4080650 IC50 = 32300.0 nM 4.49
CHEMBL4096076 IC50 = 33800.0 nM 4.47
CHEMBL4081640 IC50 > 57000.0 nM -
CHEMBL4073737 IC50 > 57000.0 nM -
CHEMBL4076264 IC50 > 57000.0 nM -
CHEMBL4066686 IC50 > 57000.0 nM -
CHEMBL4062653 IC50 > 57000.0 nM -
CHEMBL4059909 IC50 > 57000.0 nM -
CHEMBL4070504 IC50 > 57000.0 nM -
CHEMBL4094023 IC50 > 57000.0 nM -
CHEMBL4073369 IC50 > 57000.0 nM -
CHEMBL4097383 IC50 > 57000.0 nM -
CHEMBL2442491 IC50 > 57000.0 nM -
CHEMBL4060749 IC50 > 57000.0 nM -
CHEMBL4089051 IC50 > 57000.0 nM -
CHEMBL4097495 IC50 > 57000.0 nM -
CHEMBL4071354 IC50 > 57000.0 nM -
CHEMBL4090108 IC50 > 57000.0 nM -
CHEMBL4097822 IC50 > 57000.0 nM -