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Assay Detail

CHEMBL4038485

Review assay metadata, readout intent, target linkage, and publication context from the same page.

ADMET
Cytotoxicity against C57BL/6 mouse bone marrow monocytes assessed as reduction in cell viability after 72 hrs in presence of M-CSF by MTS assay
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type ADMET
Organism Mus musculus
Cell Type Bone marrow monocyte
Confidence 0 — Uncurated / Unknown
Curated By Autocuration

Target

Unchecked (CHEMBL612545)
Type UNCHECKED

Publication

Synthesis of heterocyclic ring-fused tricyclic diterpene analogs as novel inhibitors of RANKL-induced osteoclastogenesis and bone resorption.
Wei G, Wu Y, He XL, Liu T, Liu M, Luo J, Qiu WW.
Eur J Med Chem (2017) 131 : 48 -67
PubMed 28288319 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 1 4.05 4.05

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL4084109 1 4.05

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL4084109 IC50 = 88300.0 nM 4.05