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Assay Detail

CHEMBL4040223

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Functional
Antiviral activity against HBV infected in human HepG2(2.2.15) cells assessed as decrease in extracellular HBV DNA levels after 12 days by dot blot analysis
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Organism Hepatitis B virus
Confidence 1 — Organism
Curated By Autocuration

Target

Hepatitis B virus (CHEMBL613497)
Type ORGANISM
Organism Hepatitis B virus

Publication

Expanding the Antiviral Spectrum of 3-Fluoro-2-(phosphonomethoxy)propyl Acyclic Nucleoside Phosphonates: Diamyl Aspartate Amidate Prodrugs.
Luo M, Groaz E, Andrei G, Snoeck R, Kalkeri R, Ptak RG, Hartman T, Buckheit RW, Schols D, De Jonghe S, Herdewijn P.
J Med Chem (2017) 60 : 6220 -6238
PubMed 28682067 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
EC50 1 5.92 5.92

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL519667 1 5.92

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL519667 EC50 = 1200.0 nM 5.92