Assay Detail
Functional
CHEMBL4047454
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Agonist activity at human NMUR2 expressed in CHO cells assessed as increase in intracellular calcium influx after 180 secs by Fluo 4-AM dye based FLIPR assay
20
Total Activities
20
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
A potent neuromedin U receptor 2-selective alkylated peptide.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| EC50 | 20 | 8.53 | 9.70 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL4074121 | — | — | 1 | 9.70 |
| CHEMBL3356083 | — | — | 1 | 9.37 |
| CHEMBL4061906 | — | — | 1 | 9.10 |
| CHEMBL4083670 | — | — | 1 | 8.82 |
| CHEMBL4060830 | — | — | 1 | 8.74 |
| CHEMBL4092080 | — | — | 1 | 8.72 |
| CHEMBL4081819 | — | — | 1 | 8.70 |
| CHEMBL4097408 | — | — | 1 | 8.52 |
| CHEMBL4088810 | — | — | 1 | 8.48 |
| CHEMBL4073508 | — | — | 1 | 8.46 |
| CHEMBL4103826 | — | — | 1 | 8.44 |
| CHEMBL4080881 | — | — | 1 | 8.42 |
| CHEMBL4079565 | — | — | 1 | 8.38 |
| CHEMBL4105113 | — | — | 1 | 8.24 |
| CHEMBL4094147 | — | — | 1 | 8.21 |
| CHEMBL4070228 | — | — | 1 | 8.14 |
| CHEMBL4087316 | — | — | 1 | 8.08 |
| CHEMBL4067577 | — | — | 1 | 8.03 |
| CHEMBL4076016 | — | — | 1 | 8.03 |
| CHEMBL4071009 | — | — | 1 | 7.96 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL4074121 | — | EC50 | = | 0.2 | nM | 9.70 |
| CHEMBL3356083 | — | EC50 | = | 0.43 | nM | 9.37 |
| CHEMBL4061906 | — | EC50 | = | 0.8 | nM | 9.10 |
| CHEMBL4083670 | — | EC50 | = | 1.5 | nM | 8.82 |
| CHEMBL4060830 | — | EC50 | = | 1.8 | nM | 8.74 |
| CHEMBL4092080 | — | EC50 | = | 1.9 | nM | 8.72 |
| CHEMBL4081819 | — | EC50 | = | 2.0 | nM | 8.70 |
| CHEMBL4097408 | — | EC50 | = | 3.0 | nM | 8.52 |
| CHEMBL4088810 | — | EC50 | = | 3.3 | nM | 8.48 |
| CHEMBL4073508 | — | EC50 | = | 3.5 | nM | 8.46 |
| CHEMBL4103826 | — | EC50 | = | 3.6 | nM | 8.44 |
| CHEMBL4080881 | — | EC50 | = | 3.8 | nM | 8.42 |
| CHEMBL4079565 | — | EC50 | = | 4.2 | nM | 8.38 |
| CHEMBL4105113 | — | EC50 | = | 5.8 | nM | 8.24 |
| CHEMBL4094147 | — | EC50 | = | 6.2 | nM | 8.21 |
| CHEMBL4070228 | — | EC50 | = | 7.3 | nM | 8.14 |
| CHEMBL4087316 | — | EC50 | = | 8.4 | nM | 8.08 |
| CHEMBL4067577 | — | EC50 | = | 9.3 | nM | 8.03 |
| CHEMBL4076016 | — | EC50 | = | 9.4 | nM | 8.03 |
| CHEMBL4071009 | — | EC50 | = | 11.0 | nM | 7.96 |