Assay Detail
Functional
CHEMBL4047470
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Growth inhibition of human NALM16 cells after 72 hrs by CellTiter-Glo reagent based assay
16
Total Activities
16
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Cell Type | NALM16 |
| Confidence | 0 — Uncurated / Unknown |
| Curated By | Autocuration |
Publication
Diverse amide analogs of sulindac for cancer treatment and prevention.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| EC50 | 16 | 6.44 | 7.15 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL4075613 | — | — | 1 | 7.15 |
| CHEMBL4101979 | — | — | 1 | 7.01 |
| CHEMBL4061941 | — | — | 1 | 6.52 |
| CHEMBL4100716 | — | — | 1 | 6.46 |
| CHEMBL4101299 | — | — | 1 | 6.31 |
| CHEMBL4081616 | — | — | 1 | 5.89 |
| CHEMBL4072732 | — | — | 1 | 5.72 |
| CHEMBL2087735 | — | — | 1 | - |
| CHEMBL4100190 | — | — | 1 | - |
| CHEMBL4075863 | — | — | 1 | - |
| CHEMBL4093457 | — | — | 1 | - |
| CHEMBL4085818 | — | — | 1 | - |
| CHEMBL4065134 | — | — | 1 | - |
| CHEMBL4091765 | — | — | 1 | - |
| CHEMBL4083989 | — | — | 1 | - |
| CHEMBL4104867 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL4075613 | — | EC50 | = | 71.0 | nM | 7.15 |
| CHEMBL4101979 | — | EC50 | = | 97.0 | nM | 7.01 |
| CHEMBL4061941 | — | EC50 | = | 300.0 | nM | 6.52 |
| CHEMBL4100716 | — | EC50 | = | 350.0 | nM | 6.46 |
| CHEMBL4101299 | — | EC50 | = | 490.0 | nM | 6.31 |
| CHEMBL4081616 | — | EC50 | = | 1300.0 | nM | 5.89 |
| CHEMBL4072732 | — | EC50 | = | 1900.0 | nM | 5.72 |
| CHEMBL2087735 | — | EC50 | - | — | - | |
| CHEMBL4100190 | — | EC50 | - | — | - | |
| CHEMBL4075863 | — | EC50 | - | — | - | |
| CHEMBL4093457 | — | EC50 | - | — | - | |
| CHEMBL4085818 | — | EC50 | - | — | - | |
| CHEMBL4065134 | — | EC50 | - | — | - | |
| CHEMBL4091765 | — | EC50 | - | — | - | |
| CHEMBL4083989 | — | EC50 | - | — | - | |
| CHEMBL4104867 | — | EC50 | - | — | - |