Assay Detail
Functional
CHEMBL4052169
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Agonist activity at human GLP-1 receptor expressed in HEK293 cells assessed as cAMP accumulation after 30 mins by HTRF assay
21
Total Activities
21
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Cell Type | HEK293 |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
Design of Novel Exendin-Based Dual Glucagon-like Peptide 1 (GLP-1)/Glucagon Receptor Agonists.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| EC50 | 21 | 10.60 | 10.82 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL4090347 | — | — | 1 | 10.82 |
| CHEMBL4065846 | — | — | 1 | 10.76 |
| CHEMBL4069307 | — | — | 1 | 10.76 |
| CHEMBL4098545 | — | — | 1 | 10.68 |
| CHEMBL4101203 | — | — | 1 | 10.65 |
| CHEMBL4098061 | — | — | 1 | 10.65 |
| CHEMBL4060629 | — | — | 1 | 10.60 |
| CHEMBL4082505 | — | — | 1 | 10.50 |
| CHEMBL5314341 | GLUCAGON | 4.0 | 1 | 10.36 |
| CHEMBL4074468 | — | — | 1 | 10.25 |
| CHEMBL414357 | EXENATIDE | 4.0 | 1 | - |
| CHEMBL410972 | — | — | 1 | - |
| CHEMBL4524066 | — | — | 1 | - |
| CHEMBL4093458 | — | — | 1 | - |
| CHEMBL4100420 | — | — | 1 | - |
| CHEMBL4076828 | — | — | 1 | - |
| CHEMBL4080035 | — | — | 1 | - |
| CHEMBL4072029 | — | — | 1 | - |
| CHEMBL4086979 | — | — | 1 | - |
| CHEMBL4065550 | — | — | 1 | - |
| CHEMBL4095024 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL4090347 | — | EC50 | = | 0.0153 | nM | 10.82 |
| CHEMBL4065846 | — | EC50 | = | 0.0174 | nM | 10.76 |
| CHEMBL4069307 | — | EC50 | = | 0.0172 | nM | 10.76 |
| CHEMBL4098545 | — | EC50 | = | 0.0209 | nM | 10.68 |
| CHEMBL4101203 | — | EC50 | = | 0.0222 | nM | 10.65 |
| CHEMBL4098061 | — | EC50 | = | 0.0222 | nM | 10.65 |
| CHEMBL4060629 | — | EC50 | = | 0.0254 | nM | 10.60 |
| CHEMBL4082505 | — | EC50 | = | 0.0313 | nM | 10.50 |
| CHEMBL5314341 | GLUCAGON | EC50 | = | 0.0439 | nM | 10.36 |
| CHEMBL4074468 | — | EC50 | = | 0.0558 | nM | 10.25 |
| CHEMBL414357 | EXENATIDE | EC50 | = | 0.0004 | nM | - |
| CHEMBL410972 | — | EC50 | = | 0.0009 | nM | - |
| CHEMBL4524066 | — | EC50 | = | 0.0064 | nM | - |
| CHEMBL4093458 | — | EC50 | = | 0.0018 | nM | - |
| CHEMBL4100420 | — | EC50 | = | 0.0012 | nM | - |
| CHEMBL4076828 | — | EC50 | = | 0.0007 | nM | - |
| CHEMBL4080035 | — | EC50 | = | 0.0082 | nM | - |
| CHEMBL4072029 | — | EC50 | = | 0.0022 | nM | - |
| CHEMBL4086979 | — | EC50 | = | 0.0039 | nM | - |
| CHEMBL4065550 | — | EC50 | = | 0.0052 | nM | - |
| CHEMBL4095024 | — | EC50 | = | 0.0058 | nM | - |