Assay Detail
Functional
CHEMBL4052170
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Agonist activity at human glucagon receptor expressed in HEK293 cells assessed as cAMP accumulation after 30 mins by HTRF assay
21
Total Activities
21
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Cell Type | HEK293 |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
Design of Novel Exendin-Based Dual Glucagon-like Peptide 1 (GLP-1)/Glucagon Receptor Agonists.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| EC50 | 21 | 9.58 | 10.81 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL4069307 | — | — | 1 | 10.81 |
| CHEMBL4098061 | — | — | 1 | 10.58 |
| CHEMBL4076828 | — | — | 1 | 8.95 |
| CHEMBL4072029 | — | — | 1 | 8.91 |
| CHEMBL4060629 | — | — | 1 | 8.63 |
| CHEMBL5314341 | GLUCAGON | 4.0 | 1 | - |
| CHEMBL414357 | EXENATIDE | 4.0 | 1 | - |
| CHEMBL410972 | — | — | 1 | - |
| CHEMBL4524066 | — | — | 1 | - |
| CHEMBL4093458 | — | — | 1 | - |
| CHEMBL4065846 | — | — | 1 | - |
| CHEMBL4101203 | — | — | 1 | - |
| CHEMBL4074468 | — | — | 1 | - |
| CHEMBL4100420 | — | — | 1 | - |
| CHEMBL4080035 | — | — | 1 | - |
| CHEMBL4090347 | — | — | 1 | - |
| CHEMBL4086979 | — | — | 1 | - |
| CHEMBL4065550 | — | — | 1 | - |
| CHEMBL4095024 | — | — | 1 | - |
| CHEMBL4098545 | — | — | 1 | - |
| CHEMBL4082505 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL4069307 | — | EC50 | = | 0.0156 | nM | 10.81 |
| CHEMBL4098061 | — | EC50 | = | 0.0264 | nM | 10.58 |
| CHEMBL4076828 | — | EC50 | = | 1.12 | nM | 8.95 |
| CHEMBL4072029 | — | EC50 | = | 1.24 | nM | 8.91 |
| CHEMBL4060629 | — | EC50 | = | 2.32 | nM | 8.63 |
| CHEMBL5314341 | GLUCAGON | EC50 | = | 0.0004 | nM | - |
| CHEMBL414357 | EXENATIDE | EC50 | > | 1.0 | 10'8pM | - |
| CHEMBL410972 | — | EC50 | > | 0.001 | nM | - |
| CHEMBL4524066 | — | EC50 | > | 0.001 | nM | - |
| CHEMBL4093458 | — | EC50 | = | 5.8 | 10'7pM | - |
| CHEMBL4065846 | — | EC50 | = | 5.7 | 10'6pM | - |
| CHEMBL4101203 | — | EC50 | = | 1.0 | 10'7pM | - |
| CHEMBL4074468 | — | EC50 | = | 4.2 | 10'7pM | - |
| CHEMBL4100420 | — | EC50 | > | 1.0 | 10'8pM | - |
| CHEMBL4080035 | — | EC50 | = | 0.0019 | nM | - |
| CHEMBL4090347 | — | EC50 | = | 0.0089 | nM | - |
| CHEMBL4086979 | — | EC50 | = | 0.0007 | nM | - |
| CHEMBL4065550 | — | EC50 | = | 0.0062 | nM | - |
| CHEMBL4095024 | — | EC50 | = | 0.0063 | nM | - |
| CHEMBL4098545 | — | EC50 | = | 0.008 | nM | - |
| CHEMBL4082505 | — | EC50 | = | 1.7 | 10'5pM | - |