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Assay Detail

CHEMBL4052530

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Binding
Inhibition of HIV integrase strand transfer activity expressed in Escherichia coli BL21 (DE3) using 5' biotin ATGTGGAAAATCTCTAGCA primer annealed with ACTGCTAGAGATTTTCCACAT 3' Cy5 template preincubated for 10 mins followed by primer/template addition measured after 30 mins by fluorescence assay
34
Total Activities
34
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Binding
Organism Human immunodeficiency virus
Confidence 0 — Uncurated / Unknown
Curated By Autocuration

Target

Unchecked (CHEMBL612545)
Type UNCHECKED

Publication

Double-Winged 3-Hydroxypyrimidine-2,4-diones: Potent and Selective Inhibition against HIV-1 RNase H with Significant Antiviral Activity.
Vernekar SKV, Tang J, Wu B, Huber AD, Casey MC, Myshakina N, Wilson DJ, Kankanala J, Kirby KA, Parniak MA, Sarafianos SG, Wang Z.
J Med Chem (2017) 60 : 5045 -5056
PubMed 28525279 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 34 5.50 7.17

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL1229211 DOLUTEGRAVIR 4.0 1 7.17
CHEMBL4089779 1 6.85
CHEMBL4079475 1 6.64
CHEMBL254316 RALTEGRAVIR 4.0 1 6.19
CHEMBL4097509 1 5.82
CHEMBL4071378 1 5.80
CHEMBL4103071 1 5.58
CHEMBL4085120 1 5.51
CHEMBL4074881 1 5.50
CHEMBL4095319 1 5.02
CHEMBL4104008 1 4.68
CHEMBL4083483 1 4.64
CHEMBL4066264 1 4.54
CHEMBL4063811 1 4.47
CHEMBL4087618 1 4.15
CHEMBL4088773 1 -
CHEMBL4086006 1 -
CHEMBL4064482 1 -
CHEMBL4093761 1 -
CHEMBL4073058 1 -
CHEMBL4078736 1 -
CHEMBL4076618 1 -
CHEMBL4098419 1 -
CHEMBL4060013 1 -
CHEMBL4081916 1 -
CHEMBL4061749 1 -
CHEMBL4071684 1 -
CHEMBL4085394 1 -
CHEMBL4068663 1 -
CHEMBL4079744 1 -

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL1229211 DOLUTEGRAVIR IC50 = 68.0 nM 7.17
CHEMBL4089779 IC50 = 140.0 nM 6.85
CHEMBL4079475 IC50 = 230.0 nM 6.64
CHEMBL254316 RALTEGRAVIR IC50 = 650.0 nM 6.19
CHEMBL4097509 IC50 = 1500.0 nM 5.82
CHEMBL4071378 IC50 = 1600.0 nM 5.80
CHEMBL4103071 IC50 = 2600.0 nM 5.58
CHEMBL4085120 IC50 = 3100.0 nM 5.51
CHEMBL4074881 IC50 = 3200.0 nM 5.50
CHEMBL4095319 IC50 = 9500.0 nM 5.02
CHEMBL4104008 IC50 = 21000.0 nM 4.68
CHEMBL4083483 IC50 = 23000.0 nM 4.64
CHEMBL4066264 IC50 = 29000.0 nM 4.54
CHEMBL4063811 IC50 = 34000.0 nM 4.47
CHEMBL4087618 IC50 = 71000.0 nM 4.15
CHEMBL4067680 IC50 > 100000.0 nM -
CHEMBL4088905 IC50 > 100000.0 nM -
CHEMBL4101479 IC50 > 100000.0 nM -
CHEMBL4075721 IC50 > 100000.0 nM -
CHEMBL4088773 IC50 > 100000.0 nM -
CHEMBL4086006 IC50 > 100000.0 nM -
CHEMBL4064482 IC50 > 100000.0 nM -
CHEMBL4093761 IC50 > 100000.0 nM -
CHEMBL4073058 IC50 > 100000.0 nM -
CHEMBL4078736 IC50 > 100000.0 nM -
CHEMBL4076618 IC50 > 100000.0 nM -
CHEMBL4098419 IC50 > 100000.0 nM -
CHEMBL4060013 IC50 > 100000.0 nM -
CHEMBL4081916 IC50 > 100000.0 nM -
CHEMBL4061749 IC50 - -
CHEMBL4071684 IC50 - -
CHEMBL4085394 IC50 > 100000.0 nM -
CHEMBL4068663 IC50 > 100000.0 nM -
CHEMBL4079744 IC50 > 100000.0 nM -