Assay Detail
Binding
CHEMBL4054022
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Competitive inhibition of human brain mitochondria MAO-A using kynuramine as substrate by Lineweaver-Burk analysis
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Tissue | Brain |
| Subcellular | Mitochondria |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
The evaluation of 1,4-benzoquinones as inhibitors of human monoamine oxidase.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Ki | 1 | 5.02 | 5.02 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL8320 | BENZOQUINONE | — | 1 | 5.02 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL8320 | BENZOQUINONE | Ki | = | 9620.0 | nM | 5.02 |