Assay Detail
Functional
CHEMBL4056969
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Agonist activity at human Y2 receptor expressed in CHO cell membranes after 120 mins by [35S]GTPgammaS binding assay
23
Total Activities
23
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
Potent antiobesity effect of a short-length peptide YY-analogue continuously administered in mice.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| EC50 | 23 | 9.26 | 10.17 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL4090092 | — | — | 1 | 10.17 |
| CHEMBL4069205 | — | — | 1 | 9.80 |
| CHEMBL4069788 | — | — | 1 | 9.72 |
| CHEMBL4064778 | — | — | 1 | 9.70 |
| CHEMBL4094429 | — | — | 1 | 9.70 |
| CHEMBL4063306 | — | — | 1 | 9.70 |
| CHEMBL4065281 | — | — | 1 | 9.68 |
| CHEMBL439904 | — | — | 1 | 9.55 |
| CHEMBL4090786 | — | — | 1 | 9.48 |
| CHEMBL4085697 | — | — | 1 | 9.39 |
| CHEMBL4097195 | — | — | 1 | 9.38 |
| CHEMBL4090126 | — | — | 1 | 9.32 |
| CHEMBL4098787 | — | — | 1 | 9.22 |
| CHEMBL4073010 | — | — | 1 | 9.21 |
| CHEMBL4101589 | — | — | 1 | 9.18 |
| CHEMBL4075287 | — | — | 1 | 9.12 |
| CHEMBL4103628 | — | — | 1 | 9.00 |
| CHEMBL4064467 | — | — | 1 | 8.77 |
| CHEMBL4065752 | — | — | 1 | 8.74 |
| CHEMBL4071371 | — | — | 1 | 8.70 |
| CHEMBL4059729 | — | — | 1 | 8.60 |
| CHEMBL4076934 | — | — | 1 | 8.42 |
| CHEMBL4065791 | — | — | 1 | 8.36 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL4090092 | — | EC50 | = | 0.068 | nM | 10.17 |
| CHEMBL4069205 | — | EC50 | = | 0.16 | nM | 9.80 |
| CHEMBL4069788 | — | EC50 | = | 0.19 | nM | 9.72 |
| CHEMBL4064778 | — | EC50 | = | 0.2 | nM | 9.70 |
| CHEMBL4094429 | — | EC50 | = | 0.2 | nM | 9.70 |
| CHEMBL4063306 | — | EC50 | = | 0.2 | nM | 9.70 |
| CHEMBL4065281 | — | EC50 | = | 0.21 | nM | 9.68 |
| CHEMBL439904 | — | EC50 | = | 0.28 | nM | 9.55 |
| CHEMBL4090786 | — | EC50 | = | 0.33 | nM | 9.48 |
| CHEMBL4085697 | — | EC50 | = | 0.41 | nM | 9.39 |
| CHEMBL4097195 | — | EC50 | = | 0.42 | nM | 9.38 |
| CHEMBL4090126 | — | EC50 | = | 0.48 | nM | 9.32 |
| CHEMBL4098787 | — | EC50 | = | 0.6 | nM | 9.22 |
| CHEMBL4073010 | — | EC50 | = | 0.61 | nM | 9.21 |
| CHEMBL4101589 | — | EC50 | = | 0.66 | nM | 9.18 |
| CHEMBL4075287 | — | EC50 | = | 0.75 | nM | 9.12 |
| CHEMBL4103628 | — | EC50 | = | 1.0 | nM | 9.00 |
| CHEMBL4064467 | — | EC50 | = | 1.7 | nM | 8.77 |
| CHEMBL4065752 | — | EC50 | = | 1.8 | nM | 8.74 |
| CHEMBL4071371 | — | EC50 | = | 2.0 | nM | 8.70 |
| CHEMBL4059729 | — | EC50 | = | 2.5 | nM | 8.60 |
| CHEMBL4076934 | — | EC50 | = | 3.8 | nM | 8.42 |
| CHEMBL4065791 | — | EC50 | = | 4.4 | nM | 8.36 |