Assay Detail
Binding
CHEMBL4057158
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Mixed-type inhibition of Trypanosoma brucei trypanothione reductase assessed as enzyme-substrate-inhibitor complex using varying levels of trypanothione disulfide as substrate by Lineweaver-burk plot analysis
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Trypanosoma brucei |
| Confidence | 0 — Uncurated / Unknown |
| Curated By | Autocuration |
Publication
Bistacrines as potential antitrypanosomal agents.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Ki | 1 | 4.92 | 4.92 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL4066464 | — | — | 1 | 4.92 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL4066464 | — | Ki | = | 12000.0 | nM | 4.92 |