Assay Detail
Binding
CHEMBL4121510
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Displacement of [125I]alpha-dendrotoxin from rat brain voltage-gated K channel after 60 mins by scintillation counting analysis
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Rattus norvegicus |
| Confidence | 0 — Uncurated / Unknown |
| Curated By | Autocuration |
Publication
Identification and biological evaluation of thiazole-based inverse agonists of RORγt.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 1 | 9.66 | 9.66 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL4128926 | — | — | 1 | 9.66 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL4128926 | — | IC50 | = | 0.22 | nM | 9.66 |