Assay Detail
Binding
CHEMBL4123790
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Binding affinity to alpha1D adrenergic receptor (unknown origin)
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
Chiral analogues of (+)-cyclazosin as potent α1B-adrenoceptor selective antagonist.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Ki | 1 | 8.41 | 8.41 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL564481 | CYCLODOXAZOSIN | — | 1 | 8.41 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL564481 | CYCLODOXAZOSIN | Ki | = | 3.89 | nM | 8.41 |