Assay Detail
Binding
CHEMBL4134916
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Inhibition of bee venom PLA2
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Apis mellifera |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
Scalaradial Is a Potent Inhibitor of Transient Receptor Potential Melastatin 2 (TRPM2) Ion Channels.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 1 | 7.16 | 7.16 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL487005 | SCALARADIAL | — | 1 | 7.16 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL487005 | SCALARADIAL | IC50 | = | 70.0 | nM | 7.16 |