Assay Detail
Binding
CHEMBL4135162
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Inhibition of human recombinant MAO-B expressed in baculovirus infected insect cells by luminescence assay
24
Total Activities
22
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
Tying up tranylcypromine: Novel selective histone lysine specific demethylase 1 (LSD1) inhibitors.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 24 | 5.16 | 5.16 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL313833 | — | — | 1 | 5.16 |
| CHEMBL4162448 | — | — | 1 | - |
| CHEMBL4176623 | — | — | 1 | - |
| CHEMBL4166013 | — | — | 2 | - |
| CHEMBL3906257 | — | — | 1 | - |
| CHEMBL4163599 | — | — | 1 | - |
| CHEMBL4174280 | — | — | 1 | - |
| CHEMBL4171896 | — | — | 1 | - |
| CHEMBL4164024 | — | — | 1 | - |
| CHEMBL4175342 | — | — | 1 | - |
| CHEMBL4166129 | — | — | 1 | - |
| CHEMBL4161508 | — | — | 2 | - |
| CHEMBL4170367 | — | — | 1 | - |
| CHEMBL4160042 | — | — | 1 | - |
| CHEMBL4170687 | — | — | 1 | - |
| CHEMBL4170181 | — | — | 1 | - |
| CHEMBL4174674 | — | — | 1 | - |
| CHEMBL4166776 | — | — | 1 | - |
| CHEMBL4166366 | — | — | 1 | - |
| CHEMBL4166524 | — | — | 1 | - |
| CHEMBL4171003 | — | — | 1 | - |
| CHEMBL4176756 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL313833 | — | IC50 | = | 7000.0 | nM | 5.16 |
| CHEMBL4176756 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL4176623 | — | IC50 | - | — | - | |
| CHEMBL4166013 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL4161508 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL3906257 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL4166013 | — | IC50 | - | — | - | |
| CHEMBL4163599 | — | IC50 | - | — | - | |
| CHEMBL4174280 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL4171896 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL4164024 | — | IC50 | - | — | - | |
| CHEMBL4175342 | — | IC50 | - | — | - | |
| CHEMBL4161508 | — | IC50 | - | — | - | |
| CHEMBL4162448 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL4170367 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL4160042 | — | IC50 | - | — | - | |
| CHEMBL4170687 | — | IC50 | - | — | - | |
| CHEMBL4170181 | — | IC50 | - | — | - | |
| CHEMBL4174674 | — | IC50 | - | — | - | |
| CHEMBL4166776 | — | IC50 | - | — | - | |
| CHEMBL4166366 | — | IC50 | - | — | - | |
| CHEMBL4166524 | — | IC50 | - | — | - | |
| CHEMBL4171003 | — | IC50 | - | — | - | |
| CHEMBL4166129 | — | IC50 | > | 100000.0 | nM | - |