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Assay Detail

CHEMBL4135404

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Functional
Antioxidant activity assessed as H2O2 free radical scavenging activity after 1 hr by UV spectrophotometric analysis
15
Total Activities
13
Compounds Tested
2
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Confidence 0 — Uncurated / Unknown
Curated By Autocuration

Publication

Therapeutic investigations of novel indoxyl-based indolines: A drug target validation and Structure-Activity Relationship of angiotensin-converting enzyme inhibitors with cardiovascular regulation and thrombolytic potential.
Manikandan A, Moharil P, Sathishkumar M, Muñoz-Garay C, Sivakumar A.
Eur J Med Chem (2017) 141 : 417 -426
PubMed 29032034 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
Activity 12 - -
IC50 3 8.35 8.60

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL4174467 2 8.60
CHEMBL4160421 2 8.37
CHEMBL196 ASCORBIC ACID 4.0 1 8.08
CHEMBL4163389 1 -
CHEMBL4171024 1 -
CHEMBL4167651 1 -
CHEMBL4175518 1 -
CHEMBL4159339 1 -
CHEMBL4167252 1 -
CHEMBL4163798 1 -
CHEMBL4166152 1 -
CHEMBL4174072 1 -
CHEMBL4163792 1 -

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL4174467 IC50 = 2.5 nM 8.60
CHEMBL4160421 IC50 = 4.25 nM 8.37
CHEMBL196 ASCORBIC ACID IC50 = 8.25 nM 8.08
CHEMBL4163389 Activity - -
CHEMBL4171024 Activity - -
CHEMBL4160421 Activity - -
CHEMBL4167651 Activity - -
CHEMBL4175518 Activity - -
CHEMBL4159339 Activity - -
CHEMBL4167252 Activity - -
CHEMBL4174467 Activity - -
CHEMBL4163798 Activity - -
CHEMBL4166152 Activity - -
CHEMBL4174072 Activity - -
CHEMBL4163792 Activity - -