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Assay Detail

CHEMBL4136413

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Functional
Antiviral activity against Influenza A virus (A/Puerto Rico/8/1934(H1N1)) infected in MDCK cells assessed as inhibition of virus-induced cytopathic effect incubated for 48 hrs by Cell-titer-Glo assay
8
Total Activities
8
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Organism Influenza A virus
Cell Type MDCK
Confidence 1 — Organism
Curated By Intermediate

Target

Influenza A virus (CHEMBL613740)
Type ORGANISM
Organism Influenza A virus

Publication

Structure Optimization of Aloperine Derivatives as HIV-1 Entry Inhibitors.
Dang Z, Xie H, Zhu L, Zhang Q, Li Z, Huang L, Chen CH.
ACS Med Chem Lett (2017) 8 : 1199 -1203
PubMed 29152054 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
EC50 8 4.78 4.84

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL3329704 1 4.84
CHEMBL3804997 1 4.72
CHEMBL4166312 1 -
CHEMBL4173026 1 -
CHEMBL4160685 1 -
CHEMBL4176960 1 -
CHEMBL4170142 1 -
CHEMBL4159520 1 -

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL3329704 EC50 = 14500.0 nM 4.84
CHEMBL3804997 EC50 = 18900.0 nM 4.72
CHEMBL4166312 EC50 - -
CHEMBL4173026 EC50 - -
CHEMBL4160685 EC50 - -
CHEMBL4176960 EC50 - -
CHEMBL4170142 EC50 - -
CHEMBL4159520 EC50 - -