Assay Detail
Functional
CHEMBL4138495
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Antiparasite activity against Plasmodium falciparum assessed as inhibition of merozoites invasion into RBC by Geimsa staining-based assay
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Plasmodium falciparum |
| Confidence | 1 — Organism |
| Curated By | Intermediate |
Publication
Antimalarial drug discovery targeting apical membrane antigen 1.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 2 | 5.12 | 5.22 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL3596396 | — | — | 1 | 5.22 |
| CHEMBL170724 | — | — | 1 | 5.01 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL3596396 | — | IC50 | = | 6000.0 | nM | 5.22 |
| CHEMBL170724 | — | IC50 | = | 9800.0 | nM | 5.01 |