Assay Detail
Binding
CHEMBL4138820
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Inhibition of recombinant SUMO-tagged MLL1 (unknown origin) by histone methyl transferase assay
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Target
Histone-lysine N-methyltransferase 2A (CHEMBL1293299) ↗| Type | SINGLE PROTEIN |
| Organism | Homo sapiens |
Publication
Methyllysine binding domains: Structural insight and small molecule probe development.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 1 | 6.50 | 6.50 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL3798088 | — | — | 1 | 6.50 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL3798088 | — | IC50 | = | 320.0 | nM | 6.50 |