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Assay Detail

CHEMBL4139854

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Functional
Antiviral activity against CSFV infected in SK6 cells assessed as reduction of pseudo-plaque formation after 2 days by immunoperoxidase monolayer assay
11
Total Activities
11
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Organism Classical swine fever virus
Confidence 1 — Organism
Curated By Intermediate

Target

Classical swine fever virus (CHEMBL4296565)
Type ORGANISM
Organism Classical swine fever virus

Publication

Novel thioglycosyl analogs of glycosyltransferase substrates as antiviral compounds against classical swine fever virus and hepatitis C virus.
Pastuch-Gawolek G, Chaubey B, Szewczyk B, Krol E.
Eur J Med Chem (2017) 137 : 247 -262
PubMed 28601004 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 11 4.79 5.52

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL4173159 1 5.52
CHEMBL4162474 1 5.22
CHEMBL4174229 1 4.89
CHEMBL4166328 1 4.31
CHEMBL4169743 1 4.01
CHEMBL4176671 1 -
CHEMBL4162872 1 -
CHEMBL4170810 1 -
CHEMBL4159085 1 -
CHEMBL4171182 1 -
CHEMBL1259059 SOFOSBUVIR 4.0 1 -

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL4173159 IC50 = 3000.0 nM 5.52
CHEMBL4162474 IC50 = 6000.0 nM 5.22
CHEMBL4174229 IC50 = 13000.0 nM 4.89
CHEMBL4166328 IC50 = 49000.0 nM 4.31
CHEMBL4169743 IC50 = 97000.0 nM 4.01
CHEMBL4176671 IC50 = 103000.0 nM -
CHEMBL4162872 IC50 > 325000.0 nM -
CHEMBL4170810 IC50 > 299000.0 nM -
CHEMBL4159085 IC50 = 320000.0 nM -
CHEMBL4171182 IC50 = 370000.0 nM -
CHEMBL1259059 SOFOSBUVIR IC50 - -