Skip to main content
Free research Free research Free assay review with research home and workspace preview
Quick search ChEMBL 36
Assay Detail

CHEMBL4139874

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Functional
Antiviral activity against HCV infected in human Huh7-J17 cells assessed as inhibition of viral RNA replication after 72 hrs by bright-glo luciferase reporter assay
3
Total Activities
3
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Organism Hepacivirus hominis
Confidence 1 — Organism
Curated By Intermediate

Target

Hepatitis C virus (CHEMBL379)
Type ORGANISM
Organism Hepacivirus hominis

Publication

Novel thioglycosyl analogs of glycosyltransferase substrates as antiviral compounds against classical swine fever virus and hepatitis C virus.
Pastuch-Gawolek G, Chaubey B, Szewczyk B, Krol E.
Eur J Med Chem (2017) 137 : 247 -262
PubMed 28601004 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 3 6.13 7.55

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL1259059 SOFOSBUVIR 4.0 1 7.55
CHEMBL4162474 1 5.43
CHEMBL4173159 1 5.40

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL1259059 SOFOSBUVIR IC50 = 28.0 nM 7.55
CHEMBL4162474 IC50 = 3741.0 nM 5.43
CHEMBL4173159 IC50 = 4005.0 nM 5.40