Assay Detail
Binding
CHEMBL4139977
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Displacement of [3H]-diazepam from benzodiazepine receptor in rat brain membranes after 30 mins
7
Total Activities
7
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Rattus norvegicus |
| Tissue | Brain |
| Subcellular | Membrane |
| Confidence | 0 — Uncurated / Unknown |
| Curated By | Autocuration |
Publication
Azaphenothiazines - promising phenothiazine derivatives. An insight into nomenclature, synthesis, structure elucidation and biological properties.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 7 | 6.51 | 6.51 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL168400 | — | — | 1 | 6.51 |
| CHEMBL169918 | — | — | 1 | 6.51 |
| CHEMBL4169242 | — | — | 1 | 6.51 |
| CHEMBL4176425 | — | — | 1 | 6.51 |
| CHEMBL169612 | — | — | 1 | 6.51 |
| CHEMBL165820 | — | — | 1 | 6.51 |
| CHEMBL4176021 | — | — | 1 | 6.51 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL168400 | — | IC50 | = | 310.0 | nM | 6.51 |
| CHEMBL169918 | — | IC50 | = | 310.0 | nM | 6.51 |
| CHEMBL4169242 | — | IC50 | = | 310.0 | nM | 6.51 |
| CHEMBL4176425 | — | IC50 | = | 310.0 | nM | 6.51 |
| CHEMBL169612 | — | IC50 | = | 310.0 | nM | 6.51 |
| CHEMBL165820 | — | IC50 | = | 310.0 | nM | 6.51 |
| CHEMBL4176021 | — | IC50 | = | 310.0 | nM | 6.51 |