Assay Detail
Binding
CHEMBL4139985
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Inhibition of soybean lipoxygenase using linoleic acid as substrate preincubated for 5 mins followed by substrate addition measuredf after 7 mins by solution A/B solution based assay
3
Total Activities
3
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Glycine max |
| Confidence | 9 — Direct single protein target |
| Curated By | Intermediate |
Publication
Azaphenothiazines - promising phenothiazine derivatives. An insight into nomenclature, synthesis, structure elucidation and biological properties.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 3 | 4.37 | 4.67 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL437540 | — | — | 1 | 4.67 |
| CHEMBL226300 | — | — | 1 | 4.39 |
| CHEMBL4164951 | — | — | 1 | 4.06 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL437540 | — | IC50 | = | 21200.0 | nM | 4.67 |
| CHEMBL226300 | — | IC50 | = | 40700.0 | nM | 4.39 |
| CHEMBL4164951 | — | IC50 | = | 87700.0 | nM | 4.06 |