Assay Detail
Binding
CHEMBL4144178
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Inhibition of PHD2 in human Hep3B cells assessed as increase in EPO release after 24 hrs by ELISA
22
Total Activities
22
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
Discovery of JTZ-951: A HIF Prolyl Hydroxylase Inhibitor for the Treatment of Renal Anemia.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| EC50 | 22 | 4.98 | 5.38 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL4168030 | — | — | 1 | 5.38 |
| CHEMBL4174643 | — | — | 1 | 5.35 |
| CHEMBL4164403 | — | — | 1 | 5.33 |
| CHEMBL4159751 | — | — | 1 | 5.24 |
| CHEMBL4171201 | — | — | 1 | 5.24 |
| CHEMBL4175892 | — | — | 1 | 5.24 |
| CHEMBL4166742 | — | — | 1 | 5.24 |
| CHEMBL4167844 | — | — | 1 | 5.03 |
| CHEMBL4175056 | — | — | 1 | 4.92 |
| CHEMBL4167657 | — | — | 1 | 4.89 |
| CHEMBL4171371 | — | — | 1 | 4.85 |
| CHEMBL4173606 | — | — | 1 | 4.85 |
| CHEMBL4166512 | — | — | 1 | 4.82 |
| CHEMBL4162891 | — | — | 1 | 4.77 |
| CHEMBL4163070 | — | — | 1 | 4.72 |
| CHEMBL4159929 | — | — | 1 | 4.68 |
| CHEMBL426560 | — | — | 1 | 4.10 |
| CHEMBL4160770 | — | — | 1 | - |
| CHEMBL4174815 | — | — | 1 | - |
| CHEMBL4164159 | — | — | 1 | - |
| CHEMBL4159695 | — | — | 1 | - |
| CHEMBL4167612 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL4168030 | — | EC50 | = | 4200.0 | nM | 5.38 |
| CHEMBL4174643 | — | EC50 | = | 4500.0 | nM | 5.35 |
| CHEMBL4164403 | — | EC50 | = | 4700.0 | nM | 5.33 |
| CHEMBL4159751 | — | EC50 | = | 5800.0 | nM | 5.24 |
| CHEMBL4171201 | — | EC50 | = | 5800.0 | nM | 5.24 |
| CHEMBL4175892 | — | EC50 | = | 5800.0 | nM | 5.24 |
| CHEMBL4166742 | — | EC50 | = | 5700.0 | nM | 5.24 |
| CHEMBL4167844 | — | EC50 | = | 9300.0 | nM | 5.03 |
| CHEMBL4175056 | — | EC50 | = | 12000.0 | nM | 4.92 |
| CHEMBL4167657 | — | EC50 | = | 13000.0 | nM | 4.89 |
| CHEMBL4171371 | — | EC50 | = | 14000.0 | nM | 4.85 |
| CHEMBL4173606 | — | EC50 | = | 14000.0 | nM | 4.85 |
| CHEMBL4166512 | — | EC50 | = | 15000.0 | nM | 4.82 |
| CHEMBL4162891 | — | EC50 | = | 17000.0 | nM | 4.77 |
| CHEMBL4163070 | — | EC50 | = | 19000.0 | nM | 4.72 |
| CHEMBL4159929 | — | EC50 | = | 21000.0 | nM | 4.68 |
| CHEMBL426560 | — | EC50 | = | 79000.0 | nM | 4.10 |
| CHEMBL4160770 | — | EC50 | > | 30000.0 | nM | - |
| CHEMBL4174815 | — | EC50 | > | 30000.0 | nM | - |
| CHEMBL4164159 | — | EC50 | > | 30000.0 | nM | - |
| CHEMBL4159695 | — | EC50 | > | 30000.0 | nM | - |
| CHEMBL4167612 | — | EC50 | > | 30000.0 | nM | - |