Assay Detail
Binding
CHEMBL4145012
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Inhibition of rabbit IDO using tryptophan as substrate
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Oryctolagus cuniculus |
| Confidence | 0 — Uncurated / Unknown |
| Curated By | Autocuration |
Publication
Identification of Potent Indoleamine 2,3-Dioxygenase 1 (IDO1) Inhibitors Based on a Phenylimidazole Scaffold.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 2 | 4.50 | 4.52 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL4169249 | — | — | 1 | 4.52 |
| CHEMBL504816 | (L)-1-METHYLTRYPTOPHAN | — | 1 | 4.47 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL4169249 | — | IC50 | = | 30500.0 | nM | 4.52 |
| CHEMBL504816 | (L)-1-METHYLTRYPTOPHAN | IC50 | = | 34000.0 | nM | 4.47 |