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Assay Detail

CHEMBL4145104

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Binding
Binding affinity to full length human MDM4 by fluorescence polarization assay
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Binding
Organism Homo sapiens
Confidence 9 — Direct single protein target
Curated By Autocuration

Target

Protein Mdm4 (CHEMBL1255126)
Type SINGLE PROTEIN
Organism Homo sapiens

Publication

Simultaneous Targeting of RGD-Integrins and Dual Murine Double Minute Proteins in Glioblastoma Multiforme.
Merlino F, Daniele S, La Pietra V, Di Maro S, Di Leva FS, Brancaccio D, Tomassi S, Giuntini S, Cerofolini L, Fragai M, Luchinat C, Reichart F, Cavallini C, Costa B, Piccarducci R, Taliani S, Da Settimo F, Martini C, Kessler H, Novellino E, Marinelli L.
J Med Chem (2018) 61 : 4791 -4809
PubMed 29775303 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
Kd 1 8.64 8.64

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL4175039 1 8.64

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL4175039 Kd = 2.3 nM 8.64