Assay Detail
Binding
CHEMBL4145413
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Inhibition of chymotrypsin (unknown origin) by fluorescence assay
3
Total Activities
3
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Confidence | 0 — Uncurated / Unknown |
| Curated By | Autocuration |
Publication
Discovery, Synthesis, Pharmacological Profiling, and Biological Characterization of Brintonamides A-E, Novel Dual Protease and GPCR Modulators from a Marine Cyanobacterium.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 3 | 7.28 | 9.51 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL247767 | CHYMOSTATIN | — | 1 | 9.51 |
| CHEMBL4173913 | — | — | 1 | 5.05 |
| CHEMBL4168948 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL247767 | CHYMOSTATIN | IC50 | = | 0.31 | nM | 9.51 |
| CHEMBL4173913 | — | IC50 | = | 8980.0 | nM | 5.05 |
| CHEMBL4168948 | — | IC50 | > | 100000.0 | nM | - |