Assay Detail
Binding
CHEMBL4146936
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Displacement of [3H]-NMU-8 from human NMUR2 expressed in HEK293 cell membranes after 3 hrs by microscintillation counting
42
Total Activities
42
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Cell Type | HEK293 |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
Development of potent and proteolytically stable human neuromedin U receptor agonists.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 42 | 6.84 | 8.77 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL3356083 | — | — | 1 | 8.77 |
| CHEMBL4169726 | — | — | 1 | 8.70 |
| CHEMBL4177021 | — | — | 1 | 8.62 |
| CHEMBL4172552 | — | — | 1 | 8.37 |
| CHEMBL4161902 | — | — | 1 | 8.25 |
| CHEMBL4164026 | — | — | 1 | 8.00 |
| CHEMBL4166325 | — | — | 1 | 7.95 |
| CHEMBL4174679 | — | — | 1 | 7.91 |
| CHEMBL4176945 | — | — | 1 | 7.90 |
| CHEMBL4173583 | — | — | 1 | 7.89 |
| CHEMBL4169739 | — | — | 1 | 7.86 |
| CHEMBL4165538 | — | — | 1 | 7.67 |
| CHEMBL4165337 | — | — | 1 | 7.41 |
| CHEMBL3315335 | — | — | 1 | 7.36 |
| CHEMBL4175546 | — | — | 1 | 6.71 |
| CHEMBL4162868 | — | — | 1 | 6.68 |
| CHEMBL4161501 | — | — | 1 | 6.60 |
| CHEMBL4176206 | — | — | 1 | 6.58 |
| CHEMBL4169824 | — | — | 1 | 6.50 |
| CHEMBL4168753 | — | — | 1 | 6.48 |
| CHEMBL4160825 | — | — | 1 | 6.43 |
| CHEMBL4175953 | — | — | 1 | 6.37 |
| CHEMBL4159176 | — | — | 1 | 6.37 |
| CHEMBL4164680 | — | — | 1 | 6.09 |
| CHEMBL4169169 | — | — | 1 | 6.00 |
| CHEMBL4171697 | — | — | 1 | 5.99 |
| CHEMBL4164449 | — | — | 1 | 5.96 |
| CHEMBL4161037 | — | — | 1 | 5.87 |
| CHEMBL4169433 | — | — | 1 | 5.85 |
| CHEMBL4172829 | — | — | 1 | 5.81 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL3356083 | — | IC50 | = | 1.7 | nM | 8.77 |
| CHEMBL4169726 | — | IC50 | = | 2.0 | nM | 8.70 |
| CHEMBL4177021 | — | IC50 | = | 2.4 | nM | 8.62 |
| CHEMBL4172552 | — | IC50 | = | 4.3 | nM | 8.37 |
| CHEMBL4161902 | — | IC50 | = | 5.6 | nM | 8.25 |
| CHEMBL4164026 | — | IC50 | = | 9.9 | nM | 8.00 |
| CHEMBL4166325 | — | IC50 | = | 11.2 | nM | 7.95 |
| CHEMBL4174679 | — | IC50 | = | 12.3 | nM | 7.91 |
| CHEMBL4176945 | — | IC50 | = | 12.7 | nM | 7.90 |
| CHEMBL4173583 | — | IC50 | = | 13.0 | nM | 7.89 |
| CHEMBL4169739 | — | IC50 | = | 13.9 | nM | 7.86 |
| CHEMBL4165538 | — | IC50 | = | 21.4 | nM | 7.67 |
| CHEMBL4165337 | — | IC50 | = | 39.1 | nM | 7.41 |
| CHEMBL3315335 | — | IC50 | = | 43.9 | nM | 7.36 |
| CHEMBL4175546 | — | IC50 | = | 195.3 | nM | 6.71 |
| CHEMBL4162868 | — | IC50 | = | 206.9 | nM | 6.68 |
| CHEMBL4161501 | — | IC50 | = | 253.4 | nM | 6.60 |
| CHEMBL4176206 | — | IC50 | = | 261.6 | nM | 6.58 |
| CHEMBL4169824 | — | IC50 | = | 316.1 | nM | 6.50 |
| CHEMBL4168753 | — | IC50 | = | 330.8 | nM | 6.48 |
| CHEMBL4160825 | — | IC50 | = | 370.5 | nM | 6.43 |
| CHEMBL4175953 | — | IC50 | = | 424.4 | nM | 6.37 |
| CHEMBL4159176 | — | IC50 | = | 428.9 | nM | 6.37 |
| CHEMBL4164680 | — | IC50 | = | 802.9 | nM | 6.09 |
| CHEMBL4169169 | — | IC50 | = | 1010.0 | nM | 6.00 |
| CHEMBL4171697 | — | IC50 | = | 1019.0 | nM | 5.99 |
| CHEMBL4164449 | — | IC50 | = | 1089.0 | nM | 5.96 |
| CHEMBL4161037 | — | IC50 | = | 1365.0 | nM | 5.87 |
| CHEMBL4169433 | — | IC50 | = | 1403.0 | nM | 5.85 |
| CHEMBL4172829 | — | IC50 | = | 1546.0 | nM | 5.81 |
| CHEMBL4167677 | — | IC50 | = | 1649.0 | nM | 5.78 |
| CHEMBL4168351 | — | IC50 | = | 1813.0 | nM | 5.74 |
| CHEMBL4164922 | — | IC50 | = | 1857.0 | nM | 5.73 |
| CHEMBL4161095 | — | IC50 | = | 1961.0 | nM | 5.71 |
| CHEMBL4168961 | — | IC50 | = | 6132.0 | nM | 5.21 |
| CHEMBL4176146 | — | IC50 | = | 10700.0 | nM | 4.97 |
| CHEMBL4172768 | — | IC50 | - | — | - | |
| CHEMBL4172327 | — | IC50 | - | — | - | |
| CHEMBL4175315 | — | IC50 | - | — | - | |
| CHEMBL4166161 | — | IC50 | - | — | - | |
| CHEMBL4176785 | — | IC50 | - | — | - | |
| CHEMBL3356082 | — | IC50 | - | — | - |