Assay Detail
Binding
CHEMBL4149736
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Inhibition of MMP10 (unknown origin) using fluorescently-labeled substrate measured every min for 1 min
36
Total Activities
36
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
Phenotypic Screening To Discover Novel Chemical Series as Efficient Antihemorrhagic Agents.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 36 | 8.40 | 8.40 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL3417745 | — | — | 1 | 8.40 |
| CHEMBL4176163 | — | — | 1 | - |
| CHEMBL4172123 | — | — | 1 | - |
| CHEMBL4176634 | — | — | 1 | - |
| CHEMBL4162867 | — | — | 1 | - |
| CHEMBL4168363 | — | — | 1 | - |
| CHEMBL4160461 | — | — | 1 | - |
| CHEMBL4164938 | — | — | 1 | - |
| CHEMBL4175565 | — | — | 1 | - |
| CHEMBL4166420 | — | — | 1 | - |
| CHEMBL4177043 | — | — | 1 | - |
| CHEMBL4159507 | — | — | 1 | - |
| CHEMBL4167409 | — | — | 1 | - |
| CHEMBL4168773 | — | — | 1 | - |
| CHEMBL4167642 | — | — | 1 | - |
| CHEMBL4161049 | — | — | 1 | - |
| CHEMBL4171654 | — | — | 1 | - |
| CHEMBL4159737 | — | — | 1 | - |
| CHEMBL4168316 | — | — | 1 | - |
| CHEMBL4169391 | — | — | 1 | - |
| CHEMBL4162091 | — | — | 1 | - |
| CHEMBL4172782 | — | — | 1 | - |
| CHEMBL4164882 | — | — | 1 | - |
| CHEMBL4171242 | — | — | 1 | - |
| CHEMBL4163343 | — | — | 1 | - |
| CHEMBL4168955 | — | — | 1 | - |
| CHEMBL4176812 | — | — | 1 | - |
| CHEMBL4165534 | — | — | 1 | - |
| CHEMBL4173459 | — | — | 1 | - |
| CHEMBL4161466 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL3417745 | — | IC50 | = | 4.0 | nM | 8.40 |
| CHEMBL4162867 | — | IC50 | > | 10000.0 | nM | - |
| CHEMBL4167409 | — | IC50 | > | 10000.0 | nM | - |
| CHEMBL4159507 | — | IC50 | > | 10000.0 | nM | - |
| CHEMBL4177043 | — | IC50 | > | 10000.0 | nM | - |
| CHEMBL4166420 | — | IC50 | > | 10000.0 | nM | - |
| CHEMBL4175565 | — | IC50 | > | 10000.0 | nM | - |
| CHEMBL4164938 | — | IC50 | > | 10000.0 | nM | - |
| CHEMBL4160461 | — | IC50 | > | 10000.0 | nM | - |
| CHEMBL4168363 | — | IC50 | > | 10000.0 | nM | - |
| CHEMBL4168773 | — | IC50 | > | 10000.0 | nM | - |
| CHEMBL4176634 | — | IC50 | > | 10000.0 | nM | - |
| CHEMBL4172123 | — | IC50 | > | 10000.0 | nM | - |
| CHEMBL4161525 | — | IC50 | > | 10000.0 | nM | - |
| CHEMBL4171893 | — | IC50 | > | 10000.0 | nM | - |
| CHEMBL4164020 | — | IC50 | > | 10000.0 | nM | - |
| CHEMBL4166598 | — | IC50 | > | 10000.0 | nM | - |
| CHEMBL4177222 | — | IC50 | > | 10000.0 | nM | - |
| CHEMBL4170018 | — | IC50 | > | 10000.0 | nM | - |
| CHEMBL4172782 | — | IC50 | > | 10000.0 | nM | - |
| CHEMBL4161466 | — | IC50 | > | 10000.0 | nM | - |
| CHEMBL4173459 | — | IC50 | > | 10000.0 | nM | - |
| CHEMBL4165534 | — | IC50 | > | 10000.0 | nM | - |
| CHEMBL4176812 | — | IC50 | > | 10000.0 | nM | - |
| CHEMBL4168955 | — | IC50 | > | 10000.0 | nM | - |
| CHEMBL4163343 | — | IC50 | > | 10000.0 | nM | - |
| CHEMBL4171242 | — | IC50 | > | 10000.0 | nM | - |
| CHEMBL4164882 | — | IC50 | > | 10000.0 | nM | - |
| CHEMBL4167642 | — | IC50 | > | 10000.0 | nM | - |
| CHEMBL4162091 | — | IC50 | > | 10000.0 | nM | - |
| CHEMBL4169391 | — | IC50 | > | 10000.0 | nM | - |
| CHEMBL4168316 | — | IC50 | > | 10000.0 | nM | - |
| CHEMBL4159737 | — | IC50 | > | 10000.0 | nM | - |
| CHEMBL4171654 | — | IC50 | > | 10000.0 | nM | - |
| CHEMBL4176163 | — | IC50 | > | 10000.0 | nM | - |
| CHEMBL4161049 | — | IC50 | > | 10000.0 | nM | - |