Assay Detail
Binding
CHEMBL4155863
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Displacement of [125I]-CCL2 from HCMV US28 expressed in HEK293 cells after 3 hrs by gamma counting method
15
Total Activities
8
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Human betaherpesvirus 5 |
| Cell Type | HEK293 |
| Confidence | 0 — Uncurated / Unknown |
| Curated By | Autocuration |
Publication
Ligand-selective small molecule modulators of the constitutively active vGPCR US28.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 15 | 5.45 | 5.82 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL4163353 | — | — | 2 | 5.82 |
| CHEMBL4162325 | — | — | 2 | 5.68 |
| CHEMBL4172689 | — | — | 2 | 5.52 |
| CHEMBL4175646 | — | — | 2 | 5.28 |
| CHEMBL4168899 | — | — | 1 | 5.28 |
| CHEMBL4166498 | — | — | 2 | 5.02 |
| CHEMBL4169927 | — | — | 2 | - |
| CHEMBL4163068 | — | — | 2 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL4163353 | — | IC50 | = | 1520.0 | nM | 5.82 |
| CHEMBL4163353 | — | IC50 | = | 1513.56 | nM | 5.82 |
| CHEMBL4162325 | — | IC50 | = | 2110.0 | nM | 5.68 |
| CHEMBL4162325 | — | IC50 | = | 2089.3 | nM | 5.68 |
| CHEMBL4172689 | — | IC50 | = | 2990.0 | nM | 5.52 |
| CHEMBL4172689 | — | IC50 | = | 3019.95 | nM | 5.52 |
| CHEMBL4175646 | — | IC50 | = | 5260.0 | nM | 5.28 |
| CHEMBL4175646 | — | IC50 | = | 5248.07 | nM | 5.28 |
| CHEMBL4168899 | — | IC50 | = | 5290.0 | nM | 5.28 |
| CHEMBL4166498 | — | IC50 | = | 9560.0 | nM | 5.02 |
| CHEMBL4166498 | — | IC50 | = | 9549.93 | nM | 5.02 |
| CHEMBL4169927 | — | IC50 | < | 10000.0 | nM | - |
| CHEMBL4169927 | — | IC50 | > | 10000.0 | nM | - |
| CHEMBL4163068 | — | IC50 | > | 10000.0 | nM | - |
| CHEMBL4163068 | — | IC50 | < | 10000.0 | nM | - |