Assay Detail
Binding
CHEMBL4155865
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Modulation of basal activity of HCMV US28 delta300 mutant expressed in tetracyclin-induced HEK293 cells assessed as change in inositol phosphate accumulation using [3H]-myo-inositol by scintillation proximity assay
36
Total Activities
18
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Human betaherpesvirus 5 |
| Cell Type | HEK293 |
| Confidence | 0 — Uncurated / Unknown |
| Curated By | Autocuration |
Publication
Ligand-selective small molecule modulators of the constitutively active vGPCR US28.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| EC50 | 36 | 5.70 | 7.00 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL4162325 | — | — | 2 | 7.00 |
| CHEMBL4163353 | — | — | 2 | 6.74 |
| CHEMBL34166 | BERLEX COMPOUND | — | 2 | 6.10 |
| CHEMBL4166498 | — | — | 2 | 6.10 |
| CHEMBL4159986 | — | — | 2 | 5.95 |
| CHEMBL4175646 | — | — | 2 | 5.83 |
| CHEMBL4165476 | — | — | 2 | 5.82 |
| CHEMBL4162030 | — | — | 2 | 5.81 |
| CHEMBL4168899 | — | — | 2 | 5.75 |
| CHEMBL4160964 | — | — | 2 | 5.50 |
| CHEMBL4174069 | — | — | 2 | 5.32 |
| CHEMBL4176081 | — | — | 2 | 5.10 |
| CHEMBL4166806 | — | — | 2 | 5.00 |
| CHEMBL4177152 | — | — | 2 | 5.00 |
| CHEMBL4165447 | — | — | 2 | 4.70 |
| CHEMBL4167806 | — | — | 2 | - |
| CHEMBL4169309 | — | — | 2 | - |
| CHEMBL4176084 | — | — | 2 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL4162325 | — | EC50 | = | 100.0 | nM | 7.00 |
| CHEMBL4162325 | — | EC50 | = | 103.0 | nM | 6.99 |
| CHEMBL4163353 | — | EC50 | = | 182.0 | nM | 6.74 |
| CHEMBL4163353 | — | EC50 | = | 199.53 | nM | 6.70 |
| CHEMBL34166 | BERLEX COMPOUND | EC50 | = | 794.33 | nM | 6.10 |
| CHEMBL4166498 | — | EC50 | = | 794.33 | nM | 6.10 |
| CHEMBL34166 | BERLEX COMPOUND | EC50 | = | 860.0 | nM | 6.07 |
| CHEMBL4166498 | — | EC50 | = | 884.0 | nM | 6.05 |
| CHEMBL4159986 | — | EC50 | = | 1135.0 | nM | 5.95 |
| CHEMBL4159986 | — | EC50 | = | 1258.93 | nM | 5.90 |
| CHEMBL4175646 | — | EC50 | = | 1476.0 | nM | 5.83 |
| CHEMBL4165476 | — | EC50 | = | 1515.0 | nM | 5.82 |
| CHEMBL4162030 | — | EC50 | = | 1563.0 | nM | 5.81 |
| CHEMBL4175646 | — | EC50 | = | 1584.89 | nM | 5.80 |
| CHEMBL4165476 | — | EC50 | = | 1584.89 | nM | 5.80 |
| CHEMBL4162030 | — | EC50 | = | 1584.89 | nM | 5.80 |
| CHEMBL4168899 | — | EC50 | = | 1797.0 | nM | 5.75 |
| CHEMBL4168899 | — | EC50 | = | 1995.26 | nM | 5.70 |
| CHEMBL4160964 | — | EC50 | = | 3162.28 | nM | 5.50 |
| CHEMBL4160964 | — | EC50 | = | 3360.0 | nM | 5.47 |
| CHEMBL4174069 | — | EC50 | = | 4803.0 | nM | 5.32 |
| CHEMBL4174069 | — | EC50 | = | 5011.87 | nM | 5.30 |
| CHEMBL4176081 | — | EC50 | = | 7955.0 | nM | 5.10 |
| CHEMBL4176081 | — | EC50 | = | 7943.28 | nM | 5.10 |
| CHEMBL4166806 | — | EC50 | = | 9880.0 | nM | 5.00 |
| CHEMBL4166806 | — | EC50 | = | 10000.0 | nM | 5.00 |
| CHEMBL4177152 | — | EC50 | = | 10000.0 | nM | 5.00 |
| CHEMBL4177152 | — | EC50 | = | 10982.0 | nM | 4.96 |
| CHEMBL4165447 | — | EC50 | = | 19952.62 | nM | 4.70 |
| CHEMBL4165447 | — | EC50 | = | 19770.0 | nM | 4.70 |
| CHEMBL4169309 | — | EC50 | > | 10000.0 | nM | - |
| CHEMBL4169309 | — | EC50 | < | 10000.0 | nM | - |
| CHEMBL4176084 | — | EC50 | > | 10000.0 | nM | - |
| CHEMBL4176084 | — | EC50 | < | 10000.0 | nM | - |
| CHEMBL4167806 | — | EC50 | < | 10000.0 | nM | - |
| CHEMBL4167806 | — | EC50 | > | 10000.0 | nM | - |