Assay Detail
Functional
CHEMBL4155889
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Growth inhibition of human MV4-11 cells harboring FLT3-ITD after 72 hrs by Cell-Titer Glo assay
20
Total Activities
20
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Cell Type | MV4-11 |
| Confidence | 1 — Organism |
| Curated By | Intermediate |
Publication
Discovery of the selective and efficacious inhibitors of FLT3 mutations.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 20 | 7.39 | 7.80 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL4075720 | — | — | 1 | 7.80 |
| CHEMBL4163870 | — | — | 1 | 7.80 |
| CHEMBL4159478 | — | — | 1 | 7.75 |
| CHEMBL4164331 | — | — | 1 | 7.72 |
| CHEMBL4172223 | — | — | 1 | 7.58 |
| CHEMBL4160930 | — | — | 1 | 7.57 |
| CHEMBL4168869 | — | — | 1 | 7.48 |
| CHEMBL4171138 | — | — | 1 | 7.32 |
| CHEMBL4175865 | — | — | 1 | 7.28 |
| CHEMBL4167321 | — | — | 1 | 7.24 |
| CHEMBL4172658 | — | — | 1 | 7.23 |
| CHEMBL4167778 | — | — | 1 | 7.21 |
| CHEMBL4168002 | — | — | 1 | 7.21 |
| CHEMBL4160544 | — | — | 1 | 7.19 |
| CHEMBL4162003 | — | — | 1 | 7.19 |
| CHEMBL4175644 | — | — | 1 | 7.11 |
| CHEMBL4159414 | — | — | 1 | 7.01 |
| CHEMBL4164573 | — | — | 1 | - |
| CHEMBL4172459 | — | — | 1 | - |
| CHEMBL4161156 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL4075720 | — | IC50 | = | 16.0 | nM | 7.80 |
| CHEMBL4163870 | — | IC50 | = | 16.0 | nM | 7.80 |
| CHEMBL4159478 | — | IC50 | = | 18.0 | nM | 7.75 |
| CHEMBL4164331 | — | IC50 | = | 19.0 | nM | 7.72 |
| CHEMBL4172223 | — | IC50 | = | 26.0 | nM | 7.58 |
| CHEMBL4160930 | — | IC50 | = | 27.0 | nM | 7.57 |
| CHEMBL4168869 | — | IC50 | = | 33.0 | nM | 7.48 |
| CHEMBL4171138 | — | IC50 | = | 48.0 | nM | 7.32 |
| CHEMBL4175865 | — | IC50 | = | 52.0 | nM | 7.28 |
| CHEMBL4167321 | — | IC50 | = | 57.0 | nM | 7.24 |
| CHEMBL4172658 | — | IC50 | = | 59.0 | nM | 7.23 |
| CHEMBL4167778 | — | IC50 | = | 61.0 | nM | 7.21 |
| CHEMBL4168002 | — | IC50 | = | 62.0 | nM | 7.21 |
| CHEMBL4160544 | — | IC50 | = | 65.0 | nM | 7.19 |
| CHEMBL4162003 | — | IC50 | = | 65.0 | nM | 7.19 |
| CHEMBL4175644 | — | IC50 | = | 78.0 | nM | 7.11 |
| CHEMBL4159414 | — | IC50 | = | 98.0 | nM | 7.01 |
| CHEMBL4164573 | — | IC50 | - | — | - | |
| CHEMBL4172459 | — | IC50 | - | — | - | |
| CHEMBL4161156 | — | IC50 | - | — | - |