Assay Detail
Binding
CHEMBL4177774
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Binding affinity to CB1R (unknown origin)
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
Therapeutic Potential of Fatty Acid Amide Hydrolase, Monoacylglycerol Lipase, and N-Acylethanolamine Acid Amidase Inhibitors.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Ki | 2 | 6.65 | 7.30 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL15848 | ANANDAMIDE | — | 1 | 7.30 |
| CHEMBL122972 | 2-ARACHIDONOYLGLYCEROL | — | 1 | 6.00 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL15848 | ANANDAMIDE | Ki | = | 50.0 | nM | 7.30 |
| CHEMBL122972 | 2-ARACHIDONOYLGLYCEROL | Ki | = | 1000.0 | nM | 6.00 |