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Assay Detail

CHEMBL4178850

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Functional
Antiviral activity against Chikungunya virus LR2006-OPY1 infected in human Huh7.5 cells after 48 hrs by luciferase reporter gene assay
5
Total Activities
5
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Organism Chikungunya virus
Confidence 1 — Organism
Curated By Intermediate

Target

Chikungunya virus (CHEMBL4296563)
Type ORGANISM
Organism Chikungunya virus

Publication

The medicinal chemistry of Chikungunya virus.
da Silva-Júnior EF, Leoncini GO, Rodrigues ÉES, Aquino TM, Araújo-Júnior JX.
Bioorg Med Chem (2017) 25 : 4219 -4244
PubMed 28689975 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
EC50 5 5.89 6.30

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL7301 FENRETINIDE 3.0 1 6.30
CHEMBL4206476 1 5.85
CHEMBL4217232 1 5.85
CHEMBL295124 BERBERINE 4.0 1 5.72
CHEMBL4082099 1 5.72

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL7301 FENRETINIDE EC50 = 500.0 nM 6.30
CHEMBL4206476 EC50 = 1400.0 nM 5.85
CHEMBL4217232 EC50 = 1400.0 nM 5.85
CHEMBL295124 BERBERINE EC50 = 1900.0 nM 5.72
CHEMBL4082099 EC50 = 1900.0 nM 5.72