Assay Detail
Functional
CHEMBL4179033
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Agonist activity at human neuropeptide Y2 receptor expressed in CHO cell membranes assessed as stimulation of [35S]GTPgammaS binding incubated for 120 mins by liquid scintillation counting method
30
Total Activities
30
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Cell Type | CHO |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
Highly potent antiobesity effect of a short-length peptide YY analog in mice.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| EC50 | 30 | 9.59 | 9.96 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL4208191 | — | — | 1 | 9.96 |
| CHEMBL4207076 | — | — | 1 | 9.96 |
| CHEMBL4211310 | — | — | 1 | 9.89 |
| CHEMBL4206938 | — | — | 1 | 9.89 |
| CHEMBL4211953 | — | — | 1 | 9.89 |
| CHEMBL4216889 | — | — | 1 | 9.85 |
| CHEMBL4210786 | — | — | 1 | 9.82 |
| CHEMBL4202723 | — | — | 1 | 9.80 |
| CHEMBL4206417 | — | — | 1 | 9.77 |
| CHEMBL4216864 | — | — | 1 | 9.77 |
| CHEMBL4208856 | — | — | 1 | 9.77 |
| CHEMBL4207590 | — | — | 1 | 9.74 |
| CHEMBL4204797 | — | — | 1 | 9.74 |
| CHEMBL4212927 | — | — | 1 | 9.70 |
| CHEMBL4064778 | — | — | 1 | 9.70 |
| CHEMBL4205712 | — | — | 1 | 9.68 |
| CHEMBL4208023 | — | — | 1 | 9.68 |
| CHEMBL4217524 | — | — | 1 | 9.55 |
| CHEMBL4211441 | — | — | 1 | 9.55 |
| CHEMBL439904 | — | — | 1 | 9.55 |
| CHEMBL4212566 | — | — | 1 | 9.46 |
| CHEMBL4214907 | — | — | 1 | 9.40 |
| CHEMBL4213780 | — | — | 1 | 9.39 |
| CHEMBL4210343 | — | — | 1 | 9.31 |
| CHEMBL4216997 | — | — | 1 | 9.30 |
| CHEMBL4209661 | — | — | 1 | 9.30 |
| CHEMBL4203253 | — | — | 1 | 9.23 |
| CHEMBL4073010 | — | — | 1 | 9.21 |
| CHEMBL4211438 | — | — | 1 | 9.10 |
| CHEMBL4205282 | — | — | 1 | 8.70 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL4208191 | — | EC50 | = | 0.11 | nM | 9.96 |
| CHEMBL4207076 | — | EC50 | = | 0.11 | nM | 9.96 |
| CHEMBL4211310 | — | EC50 | = | 0.13 | nM | 9.89 |
| CHEMBL4206938 | — | EC50 | = | 0.13 | nM | 9.89 |
| CHEMBL4211953 | — | EC50 | = | 0.13 | nM | 9.89 |
| CHEMBL4216889 | — | EC50 | = | 0.14 | nM | 9.85 |
| CHEMBL4210786 | — | EC50 | = | 0.15 | nM | 9.82 |
| CHEMBL4202723 | — | EC50 | = | 0.16 | nM | 9.80 |
| CHEMBL4206417 | — | EC50 | = | 0.17 | nM | 9.77 |
| CHEMBL4216864 | — | EC50 | = | 0.17 | nM | 9.77 |
| CHEMBL4208856 | — | EC50 | = | 0.17 | nM | 9.77 |
| CHEMBL4207590 | — | EC50 | = | 0.18 | nM | 9.74 |
| CHEMBL4204797 | — | EC50 | = | 0.18 | nM | 9.74 |
| CHEMBL4212927 | — | EC50 | = | 0.2 | nM | 9.70 |
| CHEMBL4064778 | — | EC50 | = | 0.2 | nM | 9.70 |
| CHEMBL4205712 | — | EC50 | = | 0.21 | nM | 9.68 |
| CHEMBL4208023 | — | EC50 | = | 0.21 | nM | 9.68 |
| CHEMBL4217524 | — | EC50 | = | 0.28 | nM | 9.55 |
| CHEMBL4211441 | — | EC50 | = | 0.28 | nM | 9.55 |
| CHEMBL439904 | — | EC50 | = | 0.28 | nM | 9.55 |
| CHEMBL4212566 | — | EC50 | = | 0.35 | nM | 9.46 |
| CHEMBL4214907 | — | EC50 | = | 0.4 | nM | 9.40 |
| CHEMBL4213780 | — | EC50 | = | 0.41 | nM | 9.39 |
| CHEMBL4210343 | — | EC50 | = | 0.49 | nM | 9.31 |
| CHEMBL4216997 | — | EC50 | = | 0.5 | nM | 9.30 |
| CHEMBL4209661 | — | EC50 | = | 0.5 | nM | 9.30 |
| CHEMBL4203253 | — | EC50 | = | 0.59 | nM | 9.23 |
| CHEMBL4073010 | — | EC50 | = | 0.61 | nM | 9.21 |
| CHEMBL4211438 | — | EC50 | = | 0.8 | nM | 9.10 |
| CHEMBL4205282 | — | EC50 | = | 2.0 | nM | 8.70 |