Assay Detail
Binding
CHEMBL4184607
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Displacement of [Sar1-Ile5-Ile8]-Ang2 from Type-2 angiotensin 2 receptor AT2 in pig uterus myometrium membranes by gamma counting analysis
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Sus scrofa |
| Tissue | Myometrium |
| Subcellular | Membrane |
| Confidence | 0 — Uncurated / Unknown |
| Curated By | Autocuration |
Publication
A convenient transesterification method for synthesis of AT2 receptor ligands with improved stability in human liver microsomes.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Ki | 1 | 7.72 | 7.72 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL2086892 | — | — | 1 | 7.72 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL2086892 | — | Ki | = | 19.0 | nM | 7.72 |