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Assay Detail

CHEMBL4184974

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Functional
Antioxidant activity assessed as DPPH radical scavenging activity incubated for 30 mins under dark condition by spectrophotometric analysis
13
Total Activities
13
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Confidence 0 — Uncurated / Unknown
Curated By Autocuration

Publication

New butenolide derivatives from the marine sponge-derived fungus Aspergillus terreus.
Sun Y, Liu J, Li L, Gong C, Wang S, Yang F, Hua H, Lin H.
Bioorg Med Chem Lett (2018) 28 : 315 -318
PubMed 29295795 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 13 4.12 4.42

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL517026 1 4.42
CHEMBL3753562 1 4.07
CHEMBL600 ACETYLCYSTEINE 4.0 1 4.07
CHEMBL4097120 1 4.05
CHEMBL4068225 1 4.01
CHEMBL4203235 1 -
CHEMBL4216866 1 -
CHEMBL4213599 1 -
CHEMBL4070953 1 -
CHEMBL4079099 1 -
CHEMBL2035562 BUTYROLACTONE IV 1 -
CHEMBL4213302 1 -
CHEMBL2337339 ASPULVINONE E 1 -

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL517026 IC50 = 38000.0 nM 4.42
CHEMBL3753562 IC50 = 86000.0 nM 4.07
CHEMBL600 ACETYLCYSTEINE IC50 = 85000.0 nM 4.07
CHEMBL4097120 IC50 = 90000.0 nM 4.05
CHEMBL4068225 IC50 = 97000.0 nM 4.01
CHEMBL4203235 IC50 > 200000.0 nM -
CHEMBL4216866 IC50 > 200000.0 nM -
CHEMBL4213599 IC50 > 200000.0 nM -
CHEMBL4070953 IC50 > 200000.0 nM -
CHEMBL4079099 IC50 > 200000.0 nM -
CHEMBL2035562 BUTYROLACTONE IV IC50 = 129000.0 nM -
CHEMBL4213302 IC50 = 135000.0 nM -
CHEMBL2337339 ASPULVINONE E IC50 = 106000.0 nM -