Assay Detail
Functional
CHEMBL4186854
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Antagonist activity at P2Y1 receptor (unknown origin)
3
Total Activities
3
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
Current knowledge on the nucleotide agonists for the P2Y2 receptor.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 3 | 6.86 | 7.28 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL2112864 | — | — | 1 | 7.28 |
| CHEMBL4214232 | — | — | 1 | 6.83 |
| CHEMBL129841 | — | — | 1 | 6.48 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL2112864 | — | IC50 | = | 52.0 | nM | 7.28 |
| CHEMBL4214232 | — | IC50 | = | 148.0 | nM | 6.83 |
| CHEMBL129841 | — | IC50 | = | 330.0 | nM | 6.48 |