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Assay Detail

CHEMBL4186863

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Functional
Agonist activity at P2Y2 receptor (unknown origin) expressed in human 1321N1 cells
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Organism Homo sapiens
Confidence 9 — Direct single protein target
Curated By Autocuration

Target

P2Y purinoceptor 2 (CHEMBL4398)
Type SINGLE PROTEIN
Organism Homo sapiens

Publication

Current knowledge on the nucleotide agonists for the P2Y2 receptor.
Xu P, Feng X, Luan H, Wang J, Ge R, Li Z, Bian J.
Bioorg Med Chem (2018) 26 : 366 -375
PubMed 29254895 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
EC50 1 7.00 7.00

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL1767408 DIQUAFOSOL TETRASODIUM 4.0 1 7.00

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL1767408 DIQUAFOSOL TETRASODIUM EC50 = 100.0 nM 7.00