Skip to main content
Free research Free research Free assay review with research home and workspace preview
Quick search ChEMBL 36
Assay Detail

CHEMBL4188255

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Binding
Inhibition of PSMA (unknown origin)
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Binding
Organism Homo sapiens
Confidence 9 — Direct single protein target
Curated By Autocuration

Target

Glutamate carboxypeptidase 2 (CHEMBL1892)
Type SINGLE PROTEIN
Organism Homo sapiens

Publication

Synthesis of novel multivalent fluorescent inhibitors with high affinity to prostate cancer and their biological evaluation.
Kwon YD, Chung HJ, Lee SJ, Lee SH, Jeong BH, Kim HK.
Bioorg Med Chem Lett (2018) 28 : 572 -576
PubMed 29402740 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
Ki 1 11.00 11.00

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL510924 1 11.00

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL510924 Ki = 0.01 nM 11.00