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Assay Detail

CHEMBL4190520

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Binding
Binding affinity to HPV 18 ACATA TTTTGAACAA TTGGC LCR DNA (7559 to 7568 nucleotides) after 4 hrs by DNase I footprinting assay
3
Total Activities
3
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Binding
Organism Human papillomavirus type 18
Confidence 0 — Uncurated / Unknown
Curated By Autocuration

Target

Unchecked (CHEMBL612545)
Type UNCHECKED

Publication

Improved Antiviral Activity of a Polyamide Against High-Risk Human Papillomavirus <i>Via</i> N-Terminal Guanidinium Substitution.
Castaneda CH, Scuderi MJ, Edwards TG, Harris GD, Dupureur CM, Koeller KJ, Fisher C, Bashkin JK.
Medchemcomm (2016) 7 : 2076 -2082
PubMed 27840672 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
Kd 3 9.00 9.05

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL4217480 1 9.05
CHEMBL4213066 1 9.00
CHEMBL4205776 1 8.96

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL4217480 Kd = 0.9 nM 9.05
CHEMBL4213066 Kd = 1.0 nM 9.00
CHEMBL4205776 Kd = 1.1 nM 8.96