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Assay Detail

CHEMBL4192279

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Functional
Antiviral activity against HBV infected in human HepDES19 cells assessed as reduction in viral replication
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Organism Hepatitis B virus
Confidence 1 — Organism
Curated By Intermediate

Target

Hepatitis B virus (CHEMBL613497)
Type ORGANISM
Organism Hepatitis B virus

Publication

Synthesis of sulfamoylbenzamide derivatives as HBV capsid assembly effector.
Sari O, Boucle S, Cox BD, Ozturk T, Russell OO, Bassit L, Amblard F, Schinazi RF.
Eur J Med Chem (2017) 138 : 407 -421
PubMed 28688280 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
EC50 1 6.85 6.85

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL1730444 1 6.85

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL1730444 EC50 = 140.0 nM 6.85