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Assay Detail

CHEMBL4193441

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Functional
Antimalarial activity against synchronous culture of Plasmodium falciparum W2 ring stage infected in human erythrocytes after 48 hrs by flow cytometry
14
Total Activities
14
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Organism Plasmodium falciparum
Confidence 1 — Organism
Curated By Intermediate

Target

Plasmodium falciparum (CHEMBL364)
Type ORGANISM
Organism Plasmodium falciparum

Publication

Quinoline hybrids and their antiplasmodial and antimalarial activities.
Hu YQ, Gao C, Zhang S, Xu L, Xu Z, Feng LS, Wu X, Zhao F.
Eur J Med Chem (2017) 139 : 22 -47
PubMed 28800458 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 14 7.96 7.96

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL2316519 1 7.96
CHEMBL2316520 1 7.96
CHEMBL2316521 1 7.96
CHEMBL2316522 1 7.96
CHEMBL2316795 1 7.96
CHEMBL2316797 1 7.96
CHEMBL2316796 1 7.96
CHEMBL2316798 1 7.96
CHEMBL2316799 1 7.96
CHEMBL2316802 1 7.96
CHEMBL2316801 1 7.96
CHEMBL2316800 1 7.96
CHEMBL2316803 1 7.96
CHEMBL2316804 1 7.96

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL2316519 IC50 = 11.0 nM 7.96
CHEMBL2316520 IC50 = 11.0 nM 7.96
CHEMBL2316521 IC50 = 11.0 nM 7.96
CHEMBL2316522 IC50 = 11.0 nM 7.96
CHEMBL2316795 IC50 = 11.0 nM 7.96
CHEMBL2316797 IC50 = 11.0 nM 7.96
CHEMBL2316796 IC50 = 11.0 nM 7.96
CHEMBL2316798 IC50 = 11.0 nM 7.96
CHEMBL2316799 IC50 = 11.0 nM 7.96
CHEMBL2316802 IC50 = 11.0 nM 7.96
CHEMBL2316801 IC50 = 11.0 nM 7.96
CHEMBL2316800 IC50 = 11.0 nM 7.96
CHEMBL2316803 IC50 = 11.0 nM 7.96
CHEMBL2316804 IC50 = 11.0 nM 7.96