Assay Detail
Functional
CHEMBL4198050
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Growth inhibition of human M14/MDR1 cells after 72 hrs by MTS assay
35
Total Activities
35
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Confidence | 0 — Uncurated / Unknown |
| Curated By | Autocuration |
Publication
Synthesis and biological evaluation of indole-based UC-112 analogs as potent and selective survivin inhibitors.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 35 | 5.62 | 6.22 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL4203204 | — | — | 1 | 6.22 |
| CHEMBL4203716 | — | — | 1 | 6.16 |
| CHEMBL4218793 | — | — | 1 | 6.16 |
| CHEMBL4208078 | — | — | 1 | 6.10 |
| CHEMBL4214895 | — | — | 1 | 6.10 |
| CHEMBL4209848 | — | — | 1 | 6.05 |
| CHEMBL4212759 | — | — | 1 | 6.00 |
| CHEMBL4204974 | — | — | 1 | 6.00 |
| CHEMBL4205470 | — | — | 1 | 6.00 |
| CHEMBL4217188 | — | — | 1 | 6.00 |
| CHEMBL4215393 | — | — | 1 | 5.96 |
| CHEMBL4214373 | — | — | 1 | 5.89 |
| CHEMBL4215928 | — | — | 1 | 5.75 |
| CHEMBL4217711 | — | — | 1 | 5.72 |
| CHEMBL4210971 | — | — | 1 | 5.68 |
| CHEMBL4209981 | — | — | 1 | 5.66 |
| CHEMBL4213303 | — | — | 1 | 5.66 |
| CHEMBL4204700 | — | — | 1 | 5.55 |
| CHEMBL4207064 | — | — | 1 | 5.55 |
| CHEMBL4203443 | — | — | 1 | 5.51 |
| CHEMBL4206599 | — | — | 1 | 5.50 |
| CHEMBL4218858 | — | — | 1 | 5.48 |
| CHEMBL4202712 | — | — | 1 | 5.42 |
| CHEMBL4215109 | — | — | 1 | 5.16 |
| CHEMBL4203845 | — | — | 1 | 5.13 |
| CHEMBL4211611 | — | — | 1 | 5.10 |
| CHEMBL4211490 | — | — | 1 | 5.06 |
| CHEMBL4212145 | — | — | 1 | 4.97 |
| CHEMBL4208723 | — | — | 1 | 4.91 |
| CHEMBL4207127 | — | — | 1 | 4.91 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL4203204 | — | IC50 | = | 600.0 | nM | 6.22 |
| CHEMBL4203716 | — | IC50 | = | 700.0 | nM | 6.16 |
| CHEMBL4218793 | — | IC50 | = | 700.0 | nM | 6.16 |
| CHEMBL4208078 | — | IC50 | = | 800.0 | nM | 6.10 |
| CHEMBL4214895 | — | IC50 | = | 800.0 | nM | 6.10 |
| CHEMBL4209848 | — | IC50 | = | 900.0 | nM | 6.05 |
| CHEMBL4212759 | — | IC50 | = | 1000.0 | nM | 6.00 |
| CHEMBL4204974 | — | IC50 | = | 1000.0 | nM | 6.00 |
| CHEMBL4205470 | — | IC50 | = | 1000.0 | nM | 6.00 |
| CHEMBL4217188 | — | IC50 | = | 1000.0 | nM | 6.00 |
| CHEMBL4215393 | — | IC50 | = | 1100.0 | nM | 5.96 |
| CHEMBL4214373 | — | IC50 | = | 1300.0 | nM | 5.89 |
| CHEMBL4215928 | — | IC50 | = | 1800.0 | nM | 5.75 |
| CHEMBL4217711 | — | IC50 | = | 1900.0 | nM | 5.72 |
| CHEMBL4210971 | — | IC50 | = | 2100.0 | nM | 5.68 |
| CHEMBL4209981 | — | IC50 | = | 2200.0 | nM | 5.66 |
| CHEMBL4213303 | — | IC50 | = | 2200.0 | nM | 5.66 |
| CHEMBL4204700 | — | IC50 | = | 2800.0 | nM | 5.55 |
| CHEMBL4207064 | — | IC50 | = | 2800.0 | nM | 5.55 |
| CHEMBL4203443 | — | IC50 | = | 3100.0 | nM | 5.51 |
| CHEMBL4206599 | — | IC50 | = | 3200.0 | nM | 5.50 |
| CHEMBL4218858 | — | IC50 | = | 3300.0 | nM | 5.48 |
| CHEMBL4202712 | — | IC50 | = | 3800.0 | nM | 5.42 |
| CHEMBL4215109 | — | IC50 | = | 7000.0 | nM | 5.16 |
| CHEMBL4203845 | — | IC50 | = | 7400.0 | nM | 5.13 |
| CHEMBL4211611 | — | IC50 | = | 7900.0 | nM | 5.10 |
| CHEMBL4211490 | — | IC50 | = | 8700.0 | nM | 5.06 |
| CHEMBL4212145 | — | IC50 | = | 10700.0 | nM | 4.97 |
| CHEMBL4208723 | — | IC50 | = | 12200.0 | nM | 4.91 |
| CHEMBL4207127 | — | IC50 | = | 12200.0 | nM | 4.91 |
| CHEMBL4216591 | — | IC50 | = | 14300.0 | nM | 4.84 |
| CHEMBL4209565 | — | IC50 | - | — | - | |
| CHEMBL4207259 | — | IC50 | > | 30000.0 | nM | - |
| CHEMBL4210483 | — | IC50 | - | — | - | |
| CHEMBL4205613 | — | IC50 | - | — | - |