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Assay Detail

CHEMBL4199265

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Binding
Inhibition of adenosine A3 receptor (unknown origin)
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Binding
Organism Homo sapiens
Confidence 9 — Direct single protein target
Curated By Autocuration

Target

Adenosine receptor A3 (CHEMBL256)
Type SINGLE PROTEIN
Organism Homo sapiens

Publication

Emerging Approaches for the Identification of Protein Targets of Small Molecules - A Practitioners' Perspective.
Comess KM, McLoughlin SM, Oyer JA, Richardson PL, Stöckmann H, Vasudevan A, Warder SE.
J Med Chem (2018) 61 : 8504 -8535
PubMed 29718665 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 1 5.85 5.85

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL3769755 1 5.85

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL3769755 IC50 = 1400.0 nM 5.85